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This video by MTHFR Support™ discusses the importance of the gene CYP2C9. CYP2C9 is an important P450 enzyme that plays a role in the oxidation of xenobiotic and endogenous compounds. CYP2C9 is an enzyme involved in drug interactions. CYP2C9 is an enzyme involved in drug interactions. The following is a list of drugs involved in CYP2C9. Substrates are the substances on which an enzyme acts. An inhibitor is a gene whose presence prevents the expression of some other gene at a different locus. CYP2C9 inhibitors are CYP2C9 strong inhibitors, fluconazole, also known as diflucan. CYP2C9, moderate inhibitors. Amiodarone, also known as Cordarone. Fluvastatin, also known as Lescol. This is also true for Amentoflavone, a constituent of ginkgo biloba and St. John's wort. Sulfafenazole, an antibacterial. Valproic acid, an anticonvulsant and mood stabilizer. An inducer is a molecule that starts gene expression. CYP2C9 inducers are moderate inducers are carbamazepine, also known as Tegretol. Speak with a practitioner who understands epigenetics and Nutrigenomics at www.MTHFRSupport.org if you are concerned about CYP2C9.